ANTAGONISTI NEPEPTIDICI AI RECEPTORULUI DE TAHIKININA, PROCEDEU DE PREPARARE A ACESTORA SI COMPOZITIE FARMACEUTICA

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Interes:

Atribuire

Informații publicare:

Nr.: RO118372

Data: 30.05.2003

Inventator(i):

CHO SUNG-YONG STEPHEN [US]

CROWELL THOMAS ALAN [US]

GITTER BRUCE DONALD [US]

HIPSKIND PHILIP ARTHUR [US]

HOWBERT JAMES JEFFRY [US]

KRUSHINSKI JOSEPH HERMAN JR [US]

LOBB KAREN LYNN [US]

MUEHL BRIAN STEPHEN [US]

NIXON JAMES ARTHUR [US]

Aplicant(i):
LILLY CO ELI [US]
Clasificare:
Clasificare internationala (IPC):
A61K31/135; A61K31/165; A61K31/40; A61K31/404; A61K31/44; A61K31/4427; A61K31/4439; A61K31/445; A61K31/4468; A61K31/454; A61K31/4725; A61K31/475; A61K31/495; A61K31/496; A61K31/505; A61K31/535; A61K31/5377; A61K31/55; A61P1/00; A61P11/00; A61P11/06; A61P13/02; A61P17/06; A61P19/00; A61P19/02; A61P25/00; A61P25/18; A61P25/22; A61P25/24; A61P25/28; A61P29/00; A61P43/00; A61P9/00; C07C211/10; C07C211/27; C07C211/29; C07C211/30; C07C211/53; C07C211/58; C07C211/59; C07C217/58; C07C233/36; C07C233/44; C07C233/76; C07C233/78; C07C271/20; C07D209/12; C07D209/14; C07D209/16; C07D209/20; C07D211/58; C07D223/04; C07D233/76; C07D233/78; C07D295/12; C07D295/14; C07D295/15; C07D333/58; C07D401/12; C07D401/14; C07D403/12; C07D409/12; C07D409/14; C07D413/12

Clasificare comuna (CPC):
A61P1/00 (EP); A61P11/00 (EP); A61P11/06 (EP); A61P13/02 (EP); A61P17/06 (EP); A61P19/00 (EP); A61P19/02 (EP); A61P25/00 (EP); A61P25/18 (EP); A61P25/22 (EP); A61P25/24 (EP); A61P25/28 (EP); A61P29/00 (EP); A61P43/00 (EP); A61P9/00 (EP); C07C233/44 (EP, US); C07C233/78 (EP, US); C07C271/20 (EP, US); C07D209/14 (EP, US); C07D209/16 (EP, US); C07D401/12 (EP, US); C07D401/14 (EP, US); C07D403/12 (EP, KR, US); C07D409/12 (EP, US); C07D409/14 (EP, US)
Informații aplicație:
Nr.: RO19960000995
Data: 16.11.1994
Număr/numere prioritar(e):
US19930153847 17.11.1993 ; WO1994US13222 16.11.1994
Brevete asociate:
ATE231145; AU1098895; BR9408063; CA2176735; CN1078889; CN1141043; CO4290416; CZ141096; DE69432024; DK0729468; EP0729468; ES2189824; FI962074; HUT76269; JP3657982; JPH09505304; KR960705816; NO306210; NO962012; NZ276638; PE41395; PL180150; PL314487; PT729468; RU2140921; SG52654; TW412512; US5670499; US5684033; US6403577; US6727255; WO9514017; YU67694; ZA948926
Descriere:

Inventia se refera la o noua serie de compusi nepeptidici, antagonisti ai receptorilor de tahikinina administrati in tratamentul sau prevenirea bolilor fiziologice, la un procedeu pentru prepararea antagonistilor nepeptidici ai receptorilor de tahikinina si la o compozitie farmaceutica cu acesti compusi.