DRAJEU CU 2-METIL-4-(4-METIL-1-PIPERAZINIL)-10H-TIENO [2,3-b][1,5]BENZODIAZEPINA

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Assignment

Publication info:

No.: RO118370

Date: 30.05.2003

Inventor(s):

COCHRAN GEORGE R [US]

MORRIS TOMMY C [US]

Applicant(s):
LILLY CO ELI [US]
Classification:
International patent classification (IPC):
A61K31/55; A61K31/551; A61K47/30; A61K9/28; A61K9/30; A61K9/32; A61K9/36; A61P25/00

Cooperative patent classification (CPC):
A61K31/551 (EP); A61K9/28 (KR); A61K9/2846 (EP); A61K9/2866 (EP); A61K9/2886 (EP); A61P1/00 (EP); A61P25/00 (EP); A61P25/18 (EP); A61P25/22 (EP)
Application info:
No.: RO19970001776
Date: 22.03.1996
Priority number(s):
US19950410465 24.03.1995 ; WO1996US03918 22.03.1996
Related patents:
AP679; AR001405; AR002720; AT405606; ATA902296; ATE206924; ATE284695; AU5428096; AU696601; BG101901; BG62594; BR9607791; CA2216372; CH691217; CN1178662; CN1179102; CO4700474; CR5278; CZ296007; CZ300197; DE19681287; DE69615887; DE69634053; DK0733367; DK109097; DK1093815; DK173323; EA000938; EA199700260; EE03551; EE9700328; EG24077; EP0733367; EP1093815; ES2164837; ES2232379; FI973749; GB2313783; HU225269; HU9800410; IL117611; IS1903; IS4565; JPH11502848; KR100408172; KR19980703189; LT4350; LT97149; LU90115; LV11983; MX9707186; MY113440; NO320388; NO974363; NZ306111; OA10511; PE44997; PL188316; PL322579; PT1093815; PT733367; SE9703206; SI0733367; SI1093815; SI9620041; SK128297; SK283745; TR199701018; TW426526; UA44766; US2001018071; US2005085462; US5919485; US6190698; US6780433; US7229643; WO9629995; ZA962338
Description:

Inventia se refera la un drajeu de 2-metil-4-(4-metil-1-piperazinil)-10H-tieno[2,3-b][1,5]benzodiazepina, care contine 1...3% 2-metil-4(4-metil-1-piperazinil)-10H-tieno[2,3-b][1,5]benzodiazepina, 69,5...87,5% lactoza, 3,5...4,5% hidroxipropil celuloza, 4...6% crospovidona, 9...11% celuloza microcristalina, 0,25...1% stearat de magneziu, procentele fiind exprimate in greutate, in care tableta pentru drajefiere este acoperita cu un polimer selectat din grupul constand in hidroxipropilmetilceluloza, hidroxietil celuloza, metilhidroxi-etilceluloza, carboximetilceluloza sodica, hidroxipropil celuloza, polivinil pirolidona, copolimer al esterului dimetilaminoetilmetacrilat si de metilacrilat, copolimer de etilacrilatmetilmetacrilat, metilceluloza si etilceluloza.