SULFONAMIDE, INHIBITORI AI ASPARTIL PROTEAZEI HIV, COMPOZIŢII FARMACEUTICE CARE ÎI CONŢIN ŞI METODĂ DE TRATAMENT
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Publication info:
                            No.: RO118747
Date: 30.10.2003
                                Inventor(s):
                            
                            TUNG ROGER D [US]
MURCKO MARK A [US]
BHIDETTI GOVINDA RAO [US]
                                Applicant(s):
                            
                            VERTEX PHARMA [US]
                                                            
                                Classification:
                            
                            International patent classification (IPC):
                                    A61K31/16; A61K31/165; A61K31/17; A61K31/18; A61K31/255; A61K31/27; A61K31/325; A61K31/34; A61K31/341; A61K31/343; A61K31/35; A61K31/40; A61K31/4015; A61K31/403; A61K31/404; A61K31/41; A61K31/415; A61K31/42; A61K31/421; A61K31/4245; A61K31/425; A61K31/426; A61K31/44; A61K31/4402; A61K31/4418; A61K31/4433; A61K31/445; A61K31/47; A61K31/495; A61K31/496; A61K31/505; A61K31/535; A61K31/5375; A61K31/5377; A61K31/63; A61K38/55; A61P31/12; A61P31/18; C07C307/02; C07C307/06; C07C311/13; C07C311/18; C07C311/29; C07C311/39; C07C311/41; C07C311/46; C07D207/12; C07D207/26; C07D207/27; C07D207/28; C07D209/08; C07D209/10; C07D213/30; C07D215/48; C07D231/14; C07D239/22; C07D239/54; C07D263/24; C07D271/08; C07D277/20; C07D277/36; C07D295/12; C07D305/12; C07D307/12; C07D307/14; C07D307/20; C07D307/52; C07D307/64; C07D307/79; C07D403/12; C07D405/12; C07D409/12; C07D409/14; C07D413/12; C07D413/14; C07D417/12; C07D419/14; C07G99/00; C07K5/078; G01N33/53; G01N33/569; A61K38/00; C07D311/42
                                    Cooperative patent classification (CPC):
                                    A61P31/12 (EP); A61P31/18 (EP); C07C307/06 (EP, US); C07C311/13 (EP, US); C07C311/18 (EP, US); C07C311/29 (EP, US); C07C311/39 (EP, US); C07C311/46 (EP, US); C07D207/26 (EP, US); C07D209/08 (EP, US); C07D213/30 (EP, US); C07D213/78 (EP, US); C07D215/38 (EP, US); C07D215/48 (EP, US); C07D231/14 (EP, US); C07D239/22 (EP, US); C07D263/24 (EP, US); C07D271/08 (EP, US); C07D277/36 (EP, US); C07D307/12 (EP, US); C07D307/20 (EP, US); C07D403/12 (EP, US); C07D405/12 (EP, US); C07D409/12 (EP, US); C07D409/14 (EP, US); C07D413/12 (EP, US); C07D413/14 (EP, US); C07D417/12 (EP, US); C07K5/06139 (EP, US); A61K38/00 (EP, US); C07C2601/02 (EP, US); C07C2601/08 (EP, US); C07C2601/14 (EP, US)
                                    
                                Application info:
                            
                            No.: RO19950000479
                                
                                Date:
                                    07.09.1993
                                
                            
                                Priority number(s):
                            
                            
                                                                US19920941982
                                08.09.1992
                                ;                                                                WO1993US08458
                                07.09.1993
                                                                                            
                        
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                        Description:
Prezenta invenţie se referă la sulfonamide, inhibitori ai aspartil proteazei HIV, la compoziţiile farmaceutice care îi conţin şi la metoda de tratament. Sulfonamidele conform invenţiei sunt utilizate ca agenţi antivirali faţă de HIV-1 şi HIV-2, fiind folositori în tratamentul infecţiei HIV la un mamifer. ŕ