SULFONAMIDE, INHIBITORI AI ASPARTIL PROTEAZEI HIV, COMPOZIŢII FARMACEUTICE CARE ÎI CONŢIN ŞI METODĂ DE TRATAMENT

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Publication info:

No.: RO118747

Date: 30.10.2003

Inventor(s):

TUNG ROGER D [US]

MURCKO MARK A [US]

BHIDETTI GOVINDA RAO [US]

Applicant(s):
VERTEX PHARMA [US]
Classification:
International patent classification (IPC):
A61K31/16; A61K31/165; A61K31/17; A61K31/18; A61K31/255; A61K31/27; A61K31/325; A61K31/34; A61K31/341; A61K31/343; A61K31/35; A61K31/40; A61K31/4015; A61K31/403; A61K31/404; A61K31/41; A61K31/415; A61K31/42; A61K31/421; A61K31/4245; A61K31/425; A61K31/426; A61K31/44; A61K31/4402; A61K31/4418; A61K31/4433; A61K31/445; A61K31/47; A61K31/495; A61K31/496; A61K31/505; A61K31/535; A61K31/5375; A61K31/5377; A61K31/63; A61K38/55; A61P31/12; A61P31/18; C07C307/02; C07C307/06; C07C311/13; C07C311/18; C07C311/29; C07C311/39; C07C311/41; C07C311/46; C07D207/12; C07D207/26; C07D207/27; C07D207/28; C07D209/08; C07D209/10; C07D213/30; C07D215/48; C07D231/14; C07D239/22; C07D239/54; C07D263/24; C07D271/08; C07D277/20; C07D277/36; C07D295/12; C07D305/12; C07D307/12; C07D307/14; C07D307/20; C07D307/52; C07D307/64; C07D307/79; C07D403/12; C07D405/12; C07D409/12; C07D409/14; C07D413/12; C07D413/14; C07D417/12; C07D419/14; C07G99/00; C07K5/078; G01N33/53; G01N33/569; A61K38/00; C07D311/42

Cooperative patent classification (CPC):
A61P31/12 (EP); A61P31/18 (EP); C07C307/06 (EP, US); C07C311/13 (EP, US); C07C311/18 (EP, US); C07C311/29 (EP, US); C07C311/39 (EP, US); C07C311/46 (EP, US); C07D207/26 (EP, US); C07D209/08 (EP, US); C07D213/30 (EP, US); C07D213/78 (EP, US); C07D215/38 (EP, US); C07D215/48 (EP, US); C07D231/14 (EP, US); C07D239/22 (EP, US); C07D263/24 (EP, US); C07D271/08 (EP, US); C07D277/36 (EP, US); C07D307/12 (EP, US); C07D307/20 (EP, US); C07D403/12 (EP, US); C07D405/12 (EP, US); C07D409/12 (EP, US); C07D409/14 (EP, US); C07D413/12 (EP, US); C07D413/14 (EP, US); C07D417/12 (EP, US); C07K5/06139 (EP, US); A61K38/00 (EP, US); C07C2601/02 (EP, US); C07C2601/08 (EP, US); C07C2601/14 (EP, US)
Application info:
No.: RO19950000479
Date: 07.09.1993
Priority number(s):
US19920941982 08.09.1992 ; WO1993US08458 07.09.1993
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AP390; ATE178598; ATE241602; AU4852093; AU691160; BG62488; BG99540; BR1100824; CA2143208; CN1061339; CN1087347; CO4870779; CY2164; CZ289475; CZ58795; DE10199024; DE69324369; DE69333012; DK0659181; DK0885887; EP0659181; EP0885887; ES2131589; ES2200243; FI120685; FI951059; GEP20012579; GR3030719; HK1012631; HK1023561; HU228198; HUT71892; IL106927; IS2334; IS4068; JP3012002; JPH08501299; KR100262056; LT3302; LTIP917; LU90736; MXPA03010538; MY142901; NL300039; NO2001012; NO303444; NO950876; NZ256238; NZ314376; PH31251; PL185635; PL307858; PT885887; RU2135496; RU95109928; SG43862; SK281360; SK29395; TW254927; UA44694; US2003069222; US2006189810; US2008293727; US2010210603; US5585397; US5856353; US6372778; US7608632; WO9405639
Description:

Prezenta invenţie se referă la sulfonamide, inhibitori ai aspartil proteazei HIV, la compoziţiile farmaceutice care îi conţin şi la metoda de tratament. Sulfonamidele conform invenţiei sunt utilizate ca agenţi antivirali faţă de HIV-1 şi HIV-2, fiind folositori în tratamentul infecţiei HIV la un mamifer. ŕ

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