DERIVAŢI DE INDAZOLCARBOXAMIDE, PROCEDEU DE PREPARARE ŞI COMPOZIŢIE FARMACEUTICĂ

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Publication info:

No.: RO119617

Date: 28.01.2005

Inventor(s):

CATLOW JOHN T [US]

COHEN MARLENE L [US]

MARTINELLI MICHAEL J [US]

SCHAUS JOHN M [US]

SWANSON STEVEN P [US]

THOMPSON DENNIS C [US]

WILSON THOMAS M [US]

Applicant(s):
LILLY CO ELI [US]
Classification:
International patent classification (IPC):
A61K31/415; A61K31/4427; A61K31/445; A61K31/47; A61K31/495; A61K31/535; A61K31/55; A61P1/00; A61P25/18; A61P25/20; A61P25/28; A61P9/06; C07D231/56; C07D401/12; C07D403/00; C07D413/00

Cooperative patent classification (CPC):
A61P1/00 (EP); A61P25/00 (EP); A61P25/18 (EP); A61P25/20 (EP); A61P25/28 (EP); A61P9/00 (EP); A61P9/06 (EP); C07D231/56 (EP, US); C07D401/12 (EP, US)
Application info:
No.: RO19970001719
Date: 14.03.1996
Priority number(s):
US19950405119 16.03.1995 ; US19950485956 07.06.1995 ; WO1996US03551 14.03.1996
Related patents:
ATE203748; AU6894896; AU700842; BR9608223; CA2215359; CN1112923; CN1183041; DE69614164; DK0732333; EA000699; EA199700242; EP0732333; ES2159345; GR3037029; HU223973; HU9801386; IL117438; JPH11502230; MX9706967; NO312833; NO974221; NZ315971; PL183867; PL322362; PT732333; SK124297; SK283924; TR199700956; US5798367; US5817676; WO9633713
Description:

Prezenta invenţie se referă la derivaţi de indazolcarboxamide, la un procedeu de preparare şi la o compoziţie farmaceutică care îi conţine. Compuşii conform invenţiei au rol de agonist/antagonist ai receptorului de serotonină 5-HT4 şi prin aceasta sunt folositori în tratamentul unor boli ale sistemului nervos central, cardiovasculare sau digestive. ŕ

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