DERIVAŢI DE DOLASTATINĂ, COMPOZIŢIE FARMACEUTICĂ ŞI UTILIZAREA ACESTORA

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Interest:

Assignment

Publication info:

No.: RO119783

Date: 30.03.2005

Inventor(s):

HAUPT ANDREAS [US]

EMLING FRANZ [DE]

ROMERDAHL CYNTHIA A [US]

Applicant(s):
BASF AG [DE]
Classification:
International patent classification (IPC):
A61K38/00; A61K38/08; A61P35/00; C07K1/04; C07K5/103; C07K7/06

Cooperative patent classification (CPC):
A61K38/08 (KR); A61P35/00 (EP); C07K5/101 (EP, US); C07K7/06 (EP, KR, US); A61K38/00 (EP, US)
Application info:
No.: RO19970002254
Date: 03.06.1996
Priority number(s):
US19950472453 07.06.1995 ; WO1996EP02393 03.06.1996
Related patents:
AR003136; AR003427; ATE223431; ATE224910; AU6124196; AU6124296; AU725164; AU725170; BG102125; BG102152; BR9609423; BR9609424; CA2219818; CA2219819; CN1182153; CN1182154; CN1187198; CN1187199; CO4700526; CO4700527; CZ293682; CZ293683; CZ376397; CZ376597; DE69623472; DE69623992; DK0832104; DK0871656; EP0832104; EP0871656; ES2186783; ES2188759; HRP960257; HRP960277; HU228071; HU228073; HU9801817; HU9801910; IL122215; IL122216; JP3957751; JP4221062; JPH11504652; JPH11504653; KR100437985; KR100437986; KR19990022582; KR19990022583; MX9709146; MX9709147; MY119042; MY124487; NO317670; NO318384; NO975710; NO975711; NZ310443; NZ310444; PL185762; PL185763; PL323723; PL323726; PT832104; PT871656; RO118953; SI0832104; SI0871656; SK165397; SK282466; TR199701544; TR199701545; TW424096; TW508357; UA46775; UA46776; US5831002; WO9640751; WO9640752; ZA964710; ZA964711
Description:

Invenţia se referă la derivaţi de dolastatină şi care are structura chimică corespunzătoare formulei generale : R1R2N - CHK-CO-A-B-D-E-(F)t-K la o compoziţie farmaceutică care cuprinde o cantitate, eficientă terapeutic, de derivat de dolastatină şi un purtător acceptabil farmaceutic şi la utilizarea unui derivat de dolastatină pentru fabricarea unei compoziţii farmaceutice, pentru tratarea unei tumori la un mamifer. ŕ

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