DERIVAŢI DE EPOTILONĂ

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Assignment

Publication info:

No.: RO120340

Date: 30.12.2005

Inventor(s):

VITE GREGORY D [US]

BORZILLERI ROBERT M [US]

KIM SOONG HOON [US]

JOHNSON JAMES A [US]

Applicant(s):
BRISTOL MYERS SQUIBB CO [US]
Classification:
International patent classification (IPC):
A61K31/335; A61K31/395; A61K31/427; A61P19/00; A61P35/00; A61P43/00; C07D225/00; C07D273/00; C07D277/26; C07D313/00; C07D417/06; C07D417/08; C07D491/04; C07D491/044; C07D493/04; C07D498/04

Cooperative patent classification (CPC):
A61P19/00 (EP); A61P35/00 (EP); A61P43/00 (EP); A61P9/00 (EP); C07D225/02 (KR); C07D277/28 (KR); C07D417/06 (EP, KR, US); C07D491/04 (EP, US); C07D491/044 (EP, KR, US); C07D493/04 (EP, KR, US)
Application info:
No.: RO19990001332
Date: 16.06.1998
Priority number(s):
US19970051951P 08.07.1997 ; US19970067524P 04.12.1997 ; WO1998US12550 16.06.1998
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Description:

Prezenta invenţie se referă la derivaţi de epotilonă, cu formula generală (loc formulă), la hidraţii, solvaţii sau izomerii geometrici, optici şi stereoizomerii acestora, acceptabili din punct de vedere farmaceutic, utilizaţi la fabricarea unui medicament pentru tratamentul cancerului.