DERIVAŢI DE EPOTILONĂ
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Interest:
Assignment
Publication info:
No.: RO120340
Date: 30.12.2005
Inventor(s):
VITE GREGORY D [US]
BORZILLERI ROBERT M [US]
KIM SOONG HOON [US]
JOHNSON JAMES A [US]
Applicant(s):
BRISTOL MYERS SQUIBB CO [US]
Classification:
International patent classification (IPC):
A61K31/335; A61K31/395; A61K31/427; A61P19/00; A61P35/00; A61P43/00; C07D225/00; C07D273/00; C07D277/26; C07D313/00; C07D417/06; C07D417/08; C07D491/04; C07D491/044; C07D493/04; C07D498/04
Cooperative patent classification (CPC):
A61P19/00 (EP); A61P35/00 (EP); A61P43/00 (EP); A61P9/00 (EP); C07D225/02 (KR); C07D277/28 (KR); C07D417/06 (EP, KR, US); C07D491/04 (EP, US); C07D491/044 (EP, KR, US); C07D493/04 (EP, KR, US)
Application info:
No.: RO19990001332
Date:
16.06.1998
Priority number(s):
US19970051951P
08.07.1997
; US19970067524P
04.12.1997
; WO1998US12550
16.06.1998
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Description:
Prezenta invenţie se referă la derivaţi de epotilonă, cu formula generală (loc formulă), la hidraţii, solvaţii sau izomerii geometrici, optici şi stereoizomerii acestora, acceptabili din punct de vedere farmaceutic, utilizaţi la fabricarea unui medicament pentru tratamentul cancerului.