DERIVAŢI DE PIRIMIDINĂ ARIL ŞI HETEROCICLIL, SUBSTITUIŢI CA ANTICOAGULANŢI
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Interest:
Assignment
Publication info:
No.: RO120971
Date: 30.10.2006
Inventor(s):
DAVEY DAVID D [US]
PHILLIPS GARY B [US]
Applicant(s):
BERLEX LAB [US]
Classification:
International patent classification (IPC):
A61K31/495; A61K31/506; A61P11/00; A61P3/10; A61P31/04; A61P35/02; A61P43/00; A61P7/02; A61P9/10; C07D239/24; C07D401/14; C07D403/12; C07D403/14
Cooperative patent classification (CPC):
A61K31/506 (KR); A61P11/00 (EP); A61P3/10 (EP); A61P31/04 (EP); A61P35/02 (EP); A61P43/00 (EP); A61P7/02 (EP); A61P9/10 (EP); C07D401/14 (EP, KR, US); C07D403/12 (EP, KR, US); C07D403/14 (EP, KR, US)
Application info:
No.: RO19200100606
Date:
03.12.1999
Priority number(s):
US19980205498
04.12.1998
; WO1999US28537
03.12.1999
Related patents:
AU3107500; AU760370; BG105557; BR9915938; CA2354040; CN1329491; CZ20011932; EE200100298; EP1135131; HRP20010499; HU0104508; IL143347; JP2002531506; KR20010093799; LT2001061; LT4912; LV12783; MXPA01005656; NO20012701; NZ512104; PL348034; RU2001118466; SI20637; SK7632001; US6127376; US6372751; WO0033844; ZA200104235
Description:
Invenţia se referă la derivaţi de pirimidină aril ?i heterociclil, substituiţi, cu formulele I, II ?i III: în care Z1, Z2, R1, R2, R3, R4,R5 ?i R6 au semnificaţii bine definite, la compoziţii farmaceutice ?i la utilizarea acestora lafabricarea unui medicament anticoagulant.
