ESTERI BORONICI

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Publication info:

No.: RO122095

Date: 30.12.2008

Inventor(s):

PUTHIAPRAMPIL TOM THOMAS [IN]

SRINATH SUMITHRA [IN]

SRIDHARAN MADHAVAN [IN]

GANESH SAMBASIVAM [IN]

Applicant(s):
BIOCON LTD [IN]
Classification:
International patent classification (IPC):
A61K31/47; A61K33/22; C07B61/00; C07F5/02; C07F5/04

Cooperative patent classification (CPC):
C07F5/02 (KR); C07F5/025 (EP, US)
Application info:
No.: RO20040000728
Date: 25.02.2002
Priority number(s):
WO2002IN00032 25.02.2002
Related patents:
ATE444299; AU2002241235; BR0215602; CA2475586; CZ2004863; DK1478650; EP1478650; ES2332881; HRP20040888; HU0500125; IL163333; JP2005518427; JP4139334; KR100598079; KR20040084915; NO20043223; NZ534688; PT1478650; SK288093; SK3052004; US2005154213; US2006040898; US7238826; US7301046; WO03070733
Description:

Invenţia se referă la esteri boronici, derivaţi optici activi ai dihidroxi hexanoatului cu formula IIa (figura), care sunt utilizaţi drept intermediari pentru sinteza inhibitorilor enzimei HMG-CoA. Invenţia se referă, de asemenea, la un procedeu de obţinere a acestor compuşi.

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